2015 Antineoplastics
Overview
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Cancer treatment
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General Concepts
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Prevent DNA synthesis
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Disrupt DNA
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Antimitotics
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Immune System Modulators
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Target Proteins
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Angiogenesis Inhibitors
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Differentiating Agents
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Interfere with Hormone Function
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Treatment Strategies
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Breast cancer treatment
Prevent DNA synthesis
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Antimetabolites
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Purine analogues
/ Therapeutic uses
C. PURINE ANALOGUES :
6-MERCAPTOPURINE (6-MP), 6-THIOGUANINE (6-TG)
Therapeutic Uses
acute leukemias
6-TG
is synergistic with
CYTARABINE
search
Drug cards
Nucleotide biochemistry
Types
Nucleotide synthesis inhibitors
Folic acid analogues
Mechanism of action
Resistance
Pharmacokinetics
Therapeutic Uses
Toxicity
Leucovorin rescue
Pyrimidine analogues
Mechanism of action
Resistance
Pharmacokinetics
Therapeutic Uses
Toxicity
Purine analogues
Review of purine synthesis
Mechanism of action
Resistance
Pharmacokinetics
Therapeutic Uses
Toxicity
Tumour lysis syndrome
DNA synthesizing enzyme inhibitors
Email: Dr. Janet Fitzakerley
| ©2015 University of Minnesota Medical School Duluth | Last modified: 11-apr-15 9:39 AM